17-DMAG for Health & Longevity - Quick Reference Sheet

17-DMAG for Health & Longevity

Created on 07/18/2026 – Quick Reference based on Evidence Review created using AI4L / Opus 4.8 Audit

Experimental compound that blocks a cellular helper protein many worn-out cells rely on to survive, letting it selectively destroy aged "zombie" cells. In fast-aging mice it lowered these cells and delayed some signs of aging, but no human aging data exist. Its only human testing revealed meaningful gut, liver, and eye toxicity. Never approved; not available as a medicine. (Full Review)

Protocol

Dose
80 mg/m²
Oncology maximum without dose-limiting toxicity; no longevity dose established
Route
Intravenous
All human dosing used intravenous infusion
Schedule
Once weekly
Weekly or twice-weekly infusions; intermittent "hit-and-run" courses favored for senolytic use
Time to effect
Senescent-cell clearance
Within days
In laboratory models only
Longevity benefit
Unknown
No human timeframe ever demonstrated

Benefits

Contraindications
  • Pregnancy or breastfeeding
  • Significant liver disease (Child-Pugh B or C)
  • Significant heart disease (LVEF below ~50%)
  • Active retinal disease
  • Baseline QTc above ~470–480 ms
Key Interactions
  • Strong CYP3A4 inhibitors (ketoconazole, itraconazole, clarithromycin, ritonavir)
  • Strong CYP3A4 inducers (rifampin, carbamazepine, phenytoin)
  • High-dose acetaminophen
  • St. John's Wort, grapefruit-derived supplements
  • Other senolytics (fisetin, quercetin), high-dose green-tea catechins, kava
  • QT-prolonging drugs (amiodarone, sotalol, ondansetron)

Risk & Side Effects

  • High: Gastrointestinal toxicity; hepatotoxicity
  • Medium: Ocular toxicity; constitutional symptoms; bone-marrow suppression
  • Low: Cardiac effects; kidney and electrolyte effects
  • Speculative: Unknown risks of chronic senolytic dosing

Monitoring

Marker Target Why
ALT / AST (liver enzymes) ~10–26 U/L Detects liver injury, the key dose-limiting toxicity
Total bilirubin 0.3–1.0 mg/dL Flags impaired liver clearance
Complete blood count Neutrophils >1.5 ×10⁹/L; platelets >150 ×10⁹/L Detects bone-marrow suppression
eGFR (kidney filtration) >90 mL/min/1.73m² Kidney clearance affects drug exposure
Corrected QT interval (QTc) <440 ms Screens for heart-rhythm risk, a class concern
Left-ventricular ejection fraction (LVEF) ≥55% Confirms adequate heart pumping before use
Dilated eye (retinal) exam No retinal changes Screens for ocular toxicity of the drug class

Cadence: Liver enzymes and blood counts before each course and roughly weekly during active dosing; kidney function and electrocardiogram before each course; eye exam at baseline and promptly with any visual symptom, otherwise every 3–6 months during repeated use.

Qualitative Assessment

  • Energy and fatigue: worsening fatigue can signal toxicity rather than benefit
  • Vision: any blurring or visual change is a warning sign for retinal toxicity
  • Digestive comfort: persistent nausea, vomiting, or diarrhea indicates poor tolerance
  • General well-being: stamina and recovery between courses gauge tolerability