Dasatinib & Quercetin as a Senolytic Therapy - Quick Reference Sheet

Dasatinib & Quercetin as a Senolytic Therapy

Created on 07/23/2026 – Quick Reference based on Evidence Review created using AI4L / Opus 4.8 Audit

The first and best-known attempt to target aging by clearing worn-out cells that linger and fuel inflammation. Animal studies show improved strength, function, and survival; small early human studies lower worn-out cell counts but prove no lasting benefit. Real cautions involve blood counts, fluid balance, and the heart. Intriguing but unproven. (Full Review)

Protocol

Dose
D 100 mg + Q 1,000 mg
Once daily, taken with food
Course length
2–3 days
Consecutive treatment days per course
Frequency
Every 2 weeks to monthly
Intermittent "hit-and-run" cycling
Time to effect
Cell clearance
~11 days
Senescent-cell burden falls after one course
Physical function
~3 weeks
Mobility gains over intermittent dosing
Bone turnover
Short-term
Bone-marker changes

Benefits

Contraindications
  • Pregnancy or breastfeeding
  • Active bleeding, significant thrombocytopenia, or anticoagulation
  • History of pleural effusion, pulmonary arterial hypertension, heart failure (NYHA III–IV), or recent cardiac events
  • Prolonged QT interval
  • Severe liver impairment (Child-Pugh C)
Key Interactions
  • Strong CYP3A4 inhibitors (ketoconazole, itraconazole, clarithromycin, ritonavir)
  • Strong CYP3A4 inducers (rifampin, carbamazepine, phenytoin, St. John's Wort)
  • Other QT-prolonging drugs (amiodarone, some antipsychotics, fluoroquinolones)
  • Acid-reducing agents (omeprazole, famotidine, antacids)
  • NSAIDs (ibuprofen, naproxen)
  • Bleeding-risk supplements (fisetin, fish oil, vitamin E, ginkgo, garlic)
  • Grapefruit juice and alcohol

Risk & Side Effects

  • High: Gastrointestinal and constitutional effects
  • Medium: Cytopenias and bleeding tendency; fluid retention and pleural effusion
  • Low: Cardiac effects and QT prolongation; pulmonary arterial hypertension; drug-interaction–mediated toxicity
  • Speculative: Neurotoxicity and myelin damage; impaired tissue repair and wound healing

Monitoring

Marker Target Why
Platelet count 200–400 ×10⁹/L Detects dasatinib-related thrombocytopenia and bleeding risk
Absolute neutrophil count > 2.0 ×10⁹/L Detects neutropenia that raises infection risk
ALT / AST (liver enzymes) < 25 U/L Screens for liver stress affecting drug clearance
eGFR (kidney filtration) > 90 mL/min/1.73m² Assesses kidney function relevant to safety and disease context
hsCRP < 1.0 mg/L Tracks systemic inflammation the therapy aims to lower
IL-6 Low-normal per assay A core SASP inflammatory marker used to gauge senolytic effect
Fasting glucose / HbA1c < 90 mg/dL / < 5.4% Monitors metabolic status, relevant in metabolic and kidney contexts
QTc interval (ECG) < 440 ms Screens for QT prolongation before and during dasatinib exposure
p16INK4a (senescent-cell marker) Lower is better (research metric) Directly indexes senescent-cell burden, the therapy's target

Cadence: Blood counts and symptoms around the first one to two courses (within a few days of dosing), then reassess every 3–6 months if cycling continues; ECG at baseline and as clinically indicated in those with cardiac risk.

Qualitative Assessment

  • Energy levels and daytime fatigue
  • Physical function — walking speed, stair-climbing, grip strength
  • Breathlessness or new cough (a fluid-retention warning sign)
  • Ease of bruising or bleeding
  • General sense of recovery and well-being between cycles