Kaempferol for Health & Longevity - Quick Reference Sheet

Kaempferol for Health & Longevity

Created on 09/13/2026 – Quick Reference based on Evidence Review created using AI4L / Opus 5 – Audit

A plant pigment, recently tested in people as a concentrated supplement. Small trials show a single low oral dose lowers the oxygen and heart-rate cost of hard effort; two weeks improved sleep and daily movement. Higher dietary intake tracks with slower mental decline and fewer deaths. The safety record is thin, and one company funded every positive human trial. (Full Review)

Protocol

Core regimen
10 mg once daily
Kaempferol aglycone (the sugar-free form) orally; the dose used in every published efficacy trial
Best time of day
Morning, with a fat-containing meal
Plasma peaks near 5.8 hours; the exercise trials dosed before activity
Single versus split dosing
Single daily dose
What the trials tested and what the long absorption peak supports
Time to effect
Exercise & cardiopulmonary
Within hours
Appeared within hours of a single dose
Activity, sleep & symptoms
2–4 weeks
Activity, sleep and symptom changes emerged over this window
Cognition & mortality
Years
Any cognitive or mortality signal is an intake pattern over years

Benefits

Contraindications
  • Pregnancy and breastfeeding
  • Endocrine cancer therapy (tamoxifen, anastrozole, letrozole) during active treatment
  • Topoisomerase-II-targeted chemotherapy (etoposide, doxorubicin, mitoxantrone), or within 30 days of completion
  • Active hormone-receptor-positive breast, ovarian or endometrial cancer
  • Warfarin with an unstable or supratherapeutic international normalised ratio (above 3.5, or fluctuating by more than 1.0 between checks)
  • Diagnosed iron-deficiency anaemia (ferritin below 30 ng/mL; haemoglobin below 12.0 g/dL in women, 13.0 g/dL in men) until repleted
  • Severe hepatic impairment (Child-Pugh Class C) or advanced renal impairment (eGFR below 30 mL/min/1.73 m²)
  • Children and adolescents under 18
Key Interactions
  • CYP3A4 substrates (simvastatin, tacrolimus, ciclosporin)
  • P-glycoprotein and BCRP substrates (digoxin, nifedipine, rosuvastatin)
  • Anticoagulants and antiplatelets (warfarin, apixaban, clopidogrel, aspirin)
  • Levothyroxine and antithyroid agents (methimazole, propylthiouracil)
  • Oral iron salts (ferrous sulfate, ferrous bisglycinate) and iron-rich meals
  • Glucose-lowering agents (metformin, glimepiride, insulin)
  • Other flavonoid and polyphenol supplements (quercetin, fisetin, luteolin, myricetin, epigallocatechin gallate, curcumin)
  • High-dose fish oil and nitric-oxide-boosting supplements (beetroot nitrate)

Risk & Side Effects

  • High:
  • Medium:
  • Low: Reduced absorption of non-heme iron; blunted adaptation to endurance training
  • Speculative: Chromosomal breaks in blood-forming progenitor cells; activation of thyroid hormone and raised energy expenditure; oestrogen-receptor activity in hormone-sensitive tissue; pro-oxidant effects above the hormetic dose range; inhibition of platelet aggregation and prolonged bleeding

Monitoring

Marker Target Why
ALT / AST 10–26 U/L (women), 10–30 U/L (men) Detects hepatic stress from a concentrated extract
TSH, free T4, free T3 TSH 0.5–2.0 mIU/L; free T4 and free T3 in the upper third of range Kaempferol upregulates the enzyme activating thyroid hormone
Ferritin + transferrin saturation Ferritin 50–150 ng/mL (men, postmenopausal women), 40–100 ng/mL (menstruating women); saturation 25–35% Flavonols inhibit non-heme iron absorption
hs-CRP Below 1.0 mg/L, ideally below 0.5 mg/L Primary readout of the anti-inflammatory mechanism claimed for kaempferol
Fasting glucose + HbA1c Glucose 75–85 mg/dL; HbA1c 4.8–5.3% Glucose-lowering effect seen in rodent models; hypoglycaemia risk on sulfonylureas
eGFR + cystatin C eGFR above 90 mL/min/1.73 m² Confirms clearance capacity; excludes contraindicating renal impairment
Complete blood count No established kaempferol-specific target; track change from own baseline, anchored to haemoglobin 13.5–15.0 g/dL (men), 12.5–14.0 g/dL (women) Safety endpoint of the ongoing pharmacokinetic trial; the system implicated by the progenitor-cell findings

Cadence: Baseline, then the same panel at 6–8 weeks, 6 months and every 6–12 months thereafter; an extra thyroid check 6–8 weeks after any dose change, and an international normalised ratio within 1–2 weeks for anyone anticoagulated.

Qualitative Assessment

  • Sleep quality and sleep latency, recorded nightly from 2 weeks before starting
  • Resting heart rate on waking, and overnight heart-rate variability
  • Daily step count and spontaneous activity
  • Perceived exertion at a fixed submaximal workload
  • Energy levels, cognitive clarity and headache frequency
  • Gastrointestinal comfort