Naringenin for Health & Longevity - Quick Reference Sheet

Naringenin for Health & Longevity

Created on 07/07/2026 – Quick Reference based on Evidence Review created using AI4L / Opus 4.8 Audit

A natural compound from citrus fruit, studied as a supplement for metabolic health and healthy aging. The most developed evidence points to modestly better blood fats and reduced liver fat, plus broad anti-inflammatory and antioxidant activity. Short-term safety looks good, but most data come from animal studies; the main caution is altered processing of some medications. Promising but unproven. (Full Review)

Protocol

Dose
200 mg/day
100 mg twice daily in the human trial; practical protocols cluster in the low hundreds of mg/day (single doses of 150–900 mg tested).
Frequency
Twice daily
Short 2–3 hour half-life; splitting the daily amount into two doses sustains blood levels better than a single dose.
Timing
With meals
Absorption of this poorly water-soluble compound improves when taken with food, ideally containing some fat.
Time to effect
Blood Lipids
~4 weeks
Triglycerides, total cholesterol, and LDL fell over 4 weeks in the human trial.
Liver Fat
~4 weeks
Ultrasound-graded liver-fat severity improved over 4 weeks.
Assessment Window
1–3 months
Realistic window for judging metabolic response with consistent use.

Benefits

Contraindications
  • Pregnancy and breastfeeding
  • Hormone-sensitive cancers
  • Significant liver impairment (Child-Pugh Class B or C)
  • Narrow-therapeutic-index drugs without medical supervision (e.g., warfarin, cyclosporine)
Key Interactions
  • CYP3A4-metabolized drugs (statins, felodipine, cyclosporine, some benzodiazepines)
  • OATP-transported drugs (fexofenadine, some statins)
  • CYP1A2 and CYP2C9 drugs (theophylline, warfarin)
  • OTC drugs via the same enzymes (some antihistamines, high-intake acetaminophen)
  • Blood-sugar-lowering drugs and supplements (berberine, metformin, sulfonylureas)
  • Lipid-lowering and citrus-flavonoid supplements (bergamot, hesperidin, red yeast rice)

Risk & Side Effects

  • High:
  • Medium: Drug- and nutrient-metabolism interactions
  • Low: Gastrointestinal discomfort; potential pro-oxidant effects at high doses
  • Speculative: Estrogenic & endocrine activity; impaired adipocyte insulin signaling; unknown long-term safety at supraphysiologic doses

Monitoring

Marker Target Why
LDL cholesterol < 100 mg/dL Primary lipid target naringenin may lower
Triglycerides < 90 mg/dL Most responsive lipid marker in the human trial
HDL cholesterol > 55 mg/dL (men), > 60 mg/dL (women) May rise modestly; part of overall lipid picture
ALT < 25 U/L (men), < 20 U/L (women) Liver-cell stress marker relevant to fatty liver
AST < 25 U/L Complements ALT for liver status
GGT < 25 U/L Sensitive marker of liver and oxidative stress
Fasting glucose 75–90 mg/dL Tracks any glycemic effect
HbA1c < 5.4% Average blood sugar over ~3 months
hs-CRP < 1.0 mg/L General inflammation marker naringenin may reduce

Cadence: Baseline, then core lipid and liver markers at 4–8 weeks, then every 3–6 months; more frequently if combined with interaction-sensitive medications.

Qualitative Assessment

  • Energy levels and daytime alertness
  • Digestive comfort (watching for nausea or stomach upset)
  • Overall sense of metabolic well-being
  • Absence of any new symptoms suggesting a medication interaction