trans-Resveratrol for Health & Longevity - Quick Reference Sheet

trans-Resveratrol for Health & Longevity

Created on 08/12/2026 – Quick Reference based on Evidence Review created using AI4L / Opus 5 Audit

A plant compound from Japanese knotweed root, taken up as a longevity candidate because it appeared to switch on the cell's low-fuel machinery. In simple organisms and overfed mice that held; in people it has not translated cleanly. The most consistent human signal is better blood vessel widening. Almost none of a swallowed dose survives intact. Nothing shows longer life. (Full Review)

Protocol

Standard supplement protocol
150–500 mg once daily
trans-Resveratrol with a fat-containing meal, taken continuously
Best time of day
Morning
Bioavailability was higher after morning administration
Single versus split dosing
Once daily sufficient
The short half-life argues for splitting, but once-daily dosing was sufficient in the successful bone and vascular trials
Time to effect
Vascular measures
4–24 weeks
Nothing produces a perceptible subjective effect, so testing is the only feedback
Bone formation markers
Within 4 weeks
Bone density moved within 16 weeks
Glucose measures
4–24 weeks
Benefit appears confined to those starting with disturbed glucose handling

Benefits

Contraindications
  • Women with oestrogen-sensitive cancers, current or past (breast, endometrial), or taking tamoxifen
  • Pregnancy, breastfeeding, and children
  • Inherited or acquired bleeding disorder, full-dose anticoagulation, or within 14 days of scheduled surgery
  • Active liver disease or transaminases above three times the upper limit of normal
  • Moderate to severe kidney impairment (estimated glomerular filtration rate below 45 mL/min/1.73 m²)
Key Interactions
  • CYP3A4 substrates (simvastatin, atorvastatin, tacrolimus, apixaban)
  • CYP2C9 substrates (warfarin, phenytoin, glipizide, celecoxib)
  • CYP2D6 substrates (metoprolol, tamoxifen, fluoxetine, codeine)
  • CYP1A2 substrates (theophylline, clozapine, olanzapine, caffeine)
  • Over-the-counter medicines (aspirin, ibuprofen, naproxen, diclofenac)
  • Supplements with additive antiplatelet effects (fish oil, ginkgo, garlic extract, high-dose vitamin E, curcumin)
  • Supplements with additive metabolic or blood-pressure effects (berberine, quercetin, pterostilbene, beetroot nitrate)
  • Structured exercise training

Risk & Side Effects

  • High: Dose-Dependent Gastrointestinal Symptoms
  • Medium: Blunting of Exercise Training Adaptations; Raised Cholesterol at High Doses; Altered Clearance of Prescription Drugs; Rising Liver Enzymes at Very High Doses
  • Low: Increased Bleeding Tendency with Antithrombotic Therapy; Accelerated Brain Volume Loss; Renal Adverse Events with High-Dose Micronised Formulations
  • Speculative: Stimulation of Hormone-Sensitive Tissue; Impaired Iron Status

Monitoring

Marker Target Why
LDL-C < 80 mg/dL Detects the documented cholesterol rise at high dose
ApoB < 80 mg/dL Counts atherogenic particles more reliably than cholesterol mass
ALT 10–26 U/L (men), 8–22 U/L (women) Detects the hepatic stress signal seen at very high dose
AST 10–26 U/L Confirms an ALT rise is hepatic rather than muscular
hs-CRP < 0.5 mg/L Tracks the claimed anti-inflammatory benefit
HbA1c 4.8–5.3% Tracks the claimed glycemic benefit over three months
Fasting insulin 2–5 µIU/mL More sensitive than glucose to early insulin resistance
Ferritin 50–150 ng/mL (men), 30–120 ng/mL (women) Addresses the isolated reports of iron depletion
Bone mineral density T-score above −1.0 The only imaging endpoint with a demonstrated effect
INR 2.0–3.0 if on warfarin, otherwise 0.8–1.2 Detects the anticoagulant interaction before bleeding occurs

Cadence: Baseline before starting; lipids and liver enzymes at 12 weeks, then every 6–12 months if stable; glucose, insulin and inflammation markers at 6 months; bone density at 12–24 months; INR weekly for the first month of combined use

Qualitative Assessment

  • Digestive comfort, specifically nausea, bloating and stool frequency
  • Training response, including whether hard sessions still produce the expected week-to-week progression in strength or endurance
  • Recovery quality between hard sessions
  • Bruising and gum bleeding, as the practical proxy for altered platelet function
  • Energy stability across the day