Aviptadil for Health & Longevity - Quick Reference Sheet

Aviptadil for Health & Longevity

Created on 09/12/2026 – Quick Reference based on Evidence Review created using AI4L / Opus 5 Audit

Aviptadil is a synthetic copy of a natural signalling molecule that relaxes blood vessels and airways and quietens immune cells. Injected locally with a second drug, it restores erections in men who have failed other treatments — its strongest evidence, licensed in a few countries. For failing lungs, infusion or inhalation improves oxygen transfer briefly, but not survival. (Full Review)

Protocol

Intravenous regimen for respiratory failure
50 → 100 → 150 pmol/kg/hour
Three successive twelve-hour infusions; 600, 1,200 then 1,800 pmol/kg per day
Inhaled regimen
100 µg three times daily
Nebulised for up to 14 days
Intracavernosal regimen
25 µg with 2 mg phentolamine mesilate
Single ampoule into the lateral shaft; maximum one injection daily, three weekly
Time to effect
Erection
Within minutes
Follows intracavernosal injection
Breathlessness
Day 7
Scores separated from placebo on nebulised dosing
Oxygenation
1–3 days
From starting infusion; fades once infusion stops

Benefits

Contraindications
  • Penile implant, Peyronie's disease or cavernosal fibrosis (intracavernosal route)
  • Sickle-cell anaemia or sickle-cell trait, leukaemia, or multiple myeloma
  • Any oral or injectable anticoagulant (intracavernosal route)
  • Sexual activity medically inadvisable, including recent myocardial infarction (under 90 days) or unstable angina
  • Heart failure with left ventricular ejection fraction below 25%, or three or more vasopressors (systemic route)
  • Known hypersensitivity to aviptadil or phentolamine mesilate
  • Children and adolescents under 18 years
  • Pregnancy or breastfeeding outside a supervised protocol
Key Interactions
  • Other erectile-dysfunction drugs, including PDE5 inhibitors (sildenafil, tadalafil) and injectables (alprostadil, papaverine)
  • Nitrates and nitric-oxide donors (glyceryl trinitrate, isosorbide mononitrate)
  • Antihypertensives and vasodilators (doxazosin, amlodipine, diuretics)
  • Neprilysin inhibitors (sacubitril/valsartan)
  • Over-the-counter analgesics and antiplatelets (aspirin, ibuprofen, naproxen)
  • Over-the-counter decongestants (pseudoephedrine, phenylephrine)
  • Vasodilatory supplements (L-Arginine, L-Citrulline, beetroot nitrate, Ginkgo biloba, yohimbine)
  • Supplements affecting bleeding (fish oil, nattokinase, high-dose vitamin E, Curcuma longa extract)
  • Other interventions (vacuum erection devices, penile prosthesis, nebulised prostacyclin analogues)

Risk & Side Effects

  • High: Vasodilatory flushing, headache and dizziness
  • Medium: Secretory diarrhoea with systemic dosing; prolonged or painful erection; injection-site bruising, haematoma and penile nodules
  • Low: Infusion-related hypotension; excess serious adverse events in critical illness; cardiac events with intracavernosal use
  • Speculative: Proliferative signalling with chronic exposure; contaminants and dose error in unregulated product

Monitoring

Marker Target Why
Systolic / diastolic blood pressure 110–125 / 70–80 mmHg Detects the commonest systemic effect
Resting heart rate 55–70 bpm Tachycardia accompanies flushing
Oxygen saturation on room air 95–99% Tracks the main claimed respiratory effect
PaO₂/FiO₂ ratio Above 300 The endpoint on which trial benefit was claimed
High-sensitivity C-reactive protein (hs-CRP) Below 0.5 mg/L Anchors the anti-inflammatory claim
Interleukin-6 No established treatment target; track the change from the individual's own day-0 value The biomarker on which the sponsor trial rested
Platelet count 175–250 × 10⁹/L Governs injection-site bleeding risk
Prothrombin time / INR 0.9–1.1 Anticoagulation bars the injectable route
Serum sodium 137–142 mmol/L Detects losses from secretory diarrhoea
Serum potassium 4.0–4.5 mmol/L Diarrhoea depletes potassium fastest
Total testosterone 600–900 ng/dL Identifies a correctable cause of erectile dysfunction
Haemoglobin electrophoresis (sickle-cell screen) Negative for sickle haemoglobin Sickle disease or trait bars injectable use

Cadence: Blood pressure and heart rate continuously throughout each infusion; oxygen saturation and oxygenation ratio daily on days 1 through 3; electrolytes on day 3 if diarrhoea occurs; inflammatory markers at days 3 and 7; clinical review at 4 weeks. Injectable users are reviewed at 6 weeks, then roughly every 3 months.

Qualitative Assessment

  • Breathlessness on a standardised exertion scale
  • Flushing frequency and intensity
  • Stool frequency and consistency during systemic courses
  • Energy and exercise tolerance in the weeks after a course
  • For the injectable route, satisfaction with rigidity and duration, plus any penile pain or palpable nodules
  • Injection-related anxiety, which drives most early discontinuation